Browsing Institutt for kjemi by Subject "EGFR; Pyrrolopyrimidine; SAR; ADME; Metabolism; Erlotinib"
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Balancing potency, metabolic stability and permeability in pyrrolopyrimidine-based EGFR inhibitors
(Journal article; Peer reviewed, 2016)The present study describes our continuous effort to develop epidermal growth factor receptor (EGFR) inhibitors based on the 6-aryl-pyrrolo[2,3-d]pyrimidin-4-amine scaffold. The activity-ADME space has been evaluated by ...